Quinolone agents | Protein binding (%) | Urinary fraction (%) | Bioavailability (%) | Cmax (mg/L) | t1/2 (h) | Ref. |
---|---|---|---|---|---|---|
Ciprofloxacin | 20–40 | 40–50 | 70 | 4.3 | 4 | [6] |
Levofloxacin | 24–38 | 87 | 99 | 6.2 | 6–7 | [6] |
Sparfloxacin | 45 | 10 | 92 | 1.1 | 20 | [6] |
Trovafloxacin | 76 | 6 | 88 | 2.1 | 9.6 | [6] |
Moxifloxacin | 50 | 20 | 90 | 4.5 | 12 | [6] |
Gatifloxacin | 20 | 72 | 96 | 3.8 | 7.8 | [6] |
Avarofloxacin | 65 | 12 | 65 | 2 | 14 | [12] |
Delafloxacin | 16 | n.a. | n.a. | 10 | 12 | [39] |
Finafloxacin | n.a. | 33 | n.a. | 11 | 10 | [19] |
Zabofloxacin | n.a. | n.a. | n.a. | 2 | 8 | [27] |
Nemonoxacin | 16 | n.a. | n.a. | 5 | 15 | [40] |